Calcineurin-NFAT-DSCR1.4 signaling as druggable axis in Gαq-R183Q–driven capillary malformations

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Authors: Tong Xu, Vera Janssen, Nathalie R. Reinhard, Paula Sobrevals-Alcaraz, Robert M. van Es, A. de Haan, JF Swart, Martijn Wehrens, Hannah de Kraker, Albert Wolkerstorfer, Chantal M.A.M. van der Horst, Harmjan R. Vos
+1 more Stephan Huveneers
Cited by: 2
References: 60

Abstract

Capillary malformations (CMs) are congenital vascular lesions caused by somatic mutations in the GNAQ gene, most frequently resulting in a p.R183Q substitution in the Gαq protein in endothelial cells. However, the downstream signaling pathways by which Gαq-R183Q impairs vascular function remain poorly defined. To address this, we generated human dermal endothelial cells lacking endogenous Gαq and expressing the Gαq-R183Q mutant. Next, using SILAC-based quantitative proteomics, we mapped the Gαq-R183Q-induced endothelial phosphoproteome. These analyses identified aberrant activation of the Calcineurin-NFAT-DSCR1.4 signaling cascade as a key pathogenic feature. NFAT dysregulation and DSCR1 expression in endothelial cells were confirmed in patient-derived biopsies. Pharmacological inhibition of Calcineurin with tacrolimus partially normalized NFAT signaling in Gαq-R183Q endothelial cells. Strikingly, genetic depletion of DSCR1 in Gαq-R183Q cells fully restored Calcineurin/NFAT signaling and enabled proper endothelial migration and angiogenic sprouting, highlighting DSCR1 as a critical effector of Gαq-R183Q signaling in CMs. These findings reveal a druggable signaling circuit downstream of Gαq-R183Q that may serve as a foundation for future therapies targeting GNAQ-driven vascular malformations, including Sturge-Weber syndrome.

Fields of Study & Subjects

Vascular Malformations and Hemangiomas Signaling Pathways in Disease Dupuytren's Contracture and Treatments

Publication details

Journal / source
Angiogenesis
Publisher
Springer Science and Business Media LLC
Volume
29
Issue
2
Pages
16–16
Publication date
4 February 2026
Language
EN