Computationally guided design of N4-(2-methyl-2H-indazol-6-yl)-N2-phenylpyrimidine-2,4-diamine inhibitors of EGFR kinase targeting Cys797

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Authors: Adchata Konsue, Duangkamol Gleeson, Kiattawee Choowongkomon, Donald J.L. Jones, Pimkhuan Hannanta-anan, Robert G. Britton, M. Paul Gleeson
Cited by: 1
References: 57

Fields of Study & Subjects

Lung Cancer Treatments and Mutations Fibroblast Growth Factor Research HER2/EGFR in Cancer Research

Publication details

Journal / source
Bioorganic & Medicinal Chemistry
Publisher
Elsevier BV
Volume
134
Pages
118544–118544
Publication date
2 January 2026
Language
EN