Design, synthesis and biological evaluation of macrocyclic NTRK heterobifunctional degraders

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Authors: Corey Anderson, Jennifer Han-Chun Tsai, Oscar J. Ingham, Richard W. Deibler, Bridget T. Kreger, Prasoon Chaturvedi, Ka Ying Sharon Hung, Christopher G. Nasveschuk, James A. Henderson, Mathew E. Sowa
Cited by: 0
References: 27

Fields of Study & Subjects

Lung Cancer Treatments and Mutations Protein Degradation and Inhibitors HER2/EGFR in Cancer Research

Publication details

Journal / source
Bioorganic & Medicinal Chemistry Letters
Volume
133
Pages
130516–130516
Publication date
1 January 2026
Language
EN