Peptidomimetics Inspired by α-Synuclein or Its Chaperone αB-Crystallin Differentially Modulate α-Synuclein Aggregation

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Authors: Nicolo Bisi, Josine Marie Kothuis, Julia Kaffy, Helena Pérez Peña, Celina M. Schulz, Chiara Maria Giulia De Luca, Arianna Ciullini, Ilaria Linda Dellarole, Léa Radal, Fabio Moda, Graziella Cappelletti, Dragos Horvath
+5 more Stefano Pieraccini, Wolfgang Hoyer, Frédéric Halgand, Nicolò Tonali, Sandrine Ongeri
Cited by: 1
References: 99

Abstract

Aggregation of the α-Synuclein (αSyn) protein in neurons is responsible for synucleinopathies such as Parkinson’s disease. In healthy cells, αSyn is primarily present as monomers. Under pathological conditions, oligomers and fibrils are formed, leading to neuronal toxicity and death. No treatment prevents fatal synucleinopathies. We designed small peptidomimetics based on the structure of αSyn aggregates and on its chaperone protein αB-Crystallin. Interestingly, a relationship between the impact of peptidomimetics on the αSyn aggregation process, their sequences, and secondary conformation has been evidenced. In vitro and in cellular assays demonstrated that one compound based on αB-Crystallin was able to interfere with αSyn folding and aggregation by reducing the formation of oligomers and promoting off-pathway aggregation. The demonstration that physiological chaperone proteins can be mimicked by small peptide derivatives paves the way for new strategies to design inhibitors of amyloid protein aggregation, a hallmark of around 50 neurodegenerative and systemic amyloid diseases.

Fields of Study & Subjects

Alzheimer's disease research and treatments Heat shock proteins research Calpain Protease Function and Regulation

Publication details

Journal / source
Journal of Medicinal Chemistry
Publisher
American Chemical Society (ACS)
Volume
69
Issue
4
Pages
4059–4077
Publication date
23 January 2026
Language
EN