Synthesis and biological evaluation of novel fused pyridopyrimidine derivatives as topoisomerase I inhibitors and as potential antitumor agents: promising results in lung, ovary and gastric cancer

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Authors: Leyre Lopez-Aguileta, Endika Martín‐Encinas, Birgitta Ruth Knudsen, Cinzia Tesauro, Annalisa Schirizzi, Rosangela Montanaro, Rosalba D’Alessandro, Maria Grazia Perrone, Angela Stefanachi, Marialessandra Contino, Concepción Alonso
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Fields of Study & Subjects

Cancer therapeutics and mechanisms Quinazolinone synthesis and applications Synthesis and biological activity

Publication details

Journal / source
SSRN Electronic Journal
Publication date
1 January 2026
Document type
Preprint