What medications can cause macrocytic anemia?

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Authors: Tripdatabase
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Abstract

Numerous medications, including methotrexate, zidovudine, and nitrous oxide, have been associated with macrocytic anemia by impairing DNA synthesis or affecting vitamin metabolism.

Fields of Study & Subjects

Hematological disorders and diagnostics Folate and B Vitamins Research Pharmacovigilance and Adverse Drug Reactions

Publication details

Journal / source
Zenodo (CERN European Organization for Nuclear Research)
Publication date
15 January 2026